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Carfilzomib (CAS: 868540-17-4)
Catalog #:EBC51036
  SKU-Pack Size Availability Size Price
EBC51036-1ML In Stock 1mL(10mM in DMSO) $238.50
EBC51036-5MG In Stock 5mg $133.50
EBC51036-10MG In Stock 10mg $193.50
EBC51036-25MG In Stock 25mg $328.50
EBC51050-50MG In Stock 50mg $493.50
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Product Information
Synonym(s) PR-171, proteasome inhibitor
Chemical Name (αS)-α-[[2-(4-Morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-N-[(1S)-3-methyl-1-[[(2R)-2-methyl-2-oxiranyl]carbonyl]butyl]- L-phenylalaninamide
Application Carfilzomib is an irreversible proteasome inhibitor
CAS Number 868540-17-4
Purity ≥99.0%
Molecular Weight 719.91
Molecular Formula C₄₀H₅₇N₅O₇
SMILES CC(C)C[C@@H](C(=O)[C@]1(CO1)C)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC3=CC=CC=C3)NC(=O)CN4CCOCC4
Target & IC50 Proteasome: IC50 = 5nM
Solubility DMSO: 100 mg/mL (138.91 mM)
Preparing Stock Solutions
ConcentrationSolventMass 1 mg 5 mg 10 mg
1 mM 1.3891 ml 6.9453 ml 13.8906 ml
5 mM 0.2778 ml 1.3891 ml 2.7781 ml
10 mM 0.1389 ml 0.6945 ml 1.3891 ml
50 mM 0.0278 ml 0.1389 ml 0.2778 ml
Shipping Gel Pack
Storage Store at -20°C
Research Use For Research Use Only. Not Intended for Diagnostic Or Therapeutic Use.
Product Description

Carfilzomib (PR-171) is a next generation, irreversible and selective inhibitor of the chymotrypsin-like activity of the proteasome. It displays potent antineoplastic activity. 

Specific Protocols
>> Western Blotting Protocol >> Immunoprecipitation Protocol
>> Immunohistochemistry Protocol >> Immunofluorescence Protocol
>> Immunocytochemistry Protocol >> Flow Cytometry Protocol
>> ChIP Protocol >> ELISA Protocol
>> HPLC Protocol >> PCR Protocol
For Research Use Only, Not For Diagnostic Or Therapeutic Procedures.
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