Protein Inhibitors - PD 81723 (CAS: 132861-87-1)

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PD 81723 (CAS: 132861-87-1)

Catalog #：EBC51126

PD 81723 (CAS: 132861-87-1)

SKU-Pack Size	Availability	Size	Price
EBC51126-10MG	In Stock	10mg	€375.70
EBC51126-50MG	In Stock	50mg	€1532.70

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Product Information

Synonym(s)

PD-81723, PD81723

Chemical Name

(2-Amino-4,5-dimethyl-3-thienyl)-[3-(trifluoromethyl)phenyl]methanone

Application

PD 81723 is an allosteric potentiator that increases the functional effects of adenosine and adenosine analogs

CAS Number

132861-87-1

Purity

≥99.0%

Molecular Weight

299.31

Molecular Formula

C₁₄H₁₂F₃NOS

SMILES

CC1=C(SC(=C1C(=O)C2=CC(=CC=C2)C(F)(F)F)N)C

Solubility

DMSO: 29.93 mg/mL (100 mM)
Ethanol: 29.93 mg/mL (100 mM)

Preparing Stock Solutions

ConcentrationSolventMass	1 mg	5 mg	10 mg
1 mM	3.3410 ml	16.7051 ml	33.4102 ml
5 mM	0.6682 ml	3.3410 ml	6.6820 ml
10 mM	0.3341 ml	1.6705 ml	3.3410 ml
50 mM	0.0668 ml	0.3341 ml	0.6682 ml

Shipping

Gel Pack

Storage

Store at -20°C

Research Use

For Research Use Only. Not Intended for Diagnostic Or Therapeutic Use.

Product Description

PD 81723 is an allosteric potentiator at Adenosine A1-R that acts via agonist-dependent and independent mechanisms. PD 81723 enhances the functional effects of adenosine and adenosine analogs. This compound also inhibits basal and forskolin-stimulated A cyclase (adenylyl cyclase, AC) activity in Adensosine A1-R expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of A cyclase (adenylyl cyclase, AC).

Specific Protocols

>>	Western Blotting Protocol	>>	Immunoprecipitation Protocol
>>	Immunohistochemistry Protocol	>>	Immunofluorescence Protocol
>>	Immunocytochemistry Protocol	>>	Flow Cytometry Protocol
>>	ChIP Protocol	>>	ELISA Protocol
>>	HPLC Protocol	>>	PCR Protocol