Protein Agonists, Antagonists and Activators

G-15 (CAS: 1161002-05-6)

Catalog #：EBC51099

G-15 (CAS: 1161002-05-6)

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Product Information

Synonym(s)

AC1LMJHT, CTK8E6722, ZINC00871833

Chemical Name

(3aR,4R,9bS)-4-(6-bromobenzo[d][1,3]dioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline

Application

G-15 is a cell-permeable non-steroidal antagonist of GPER

CAS Number

1161002-05-6

Purity

≥99.0%

Molecular Weight

370.24

Molecular Formula

C₁₉H₁₆BrNO₂

SMILES

BrC1=CC2=C(OCO2)C=C1[C@@H]3NC(C=CC=C4)=C4[C@@]5([H])[C@]3([H])CC=C5

Target & IC50

GPER/GPR30

Solubility

DMSO: 41.67 mg/mL (112.55 mM)

Preparing Stock Solutions

Shipping

Gel Pack

Storage

Store at -20°C

Research Use

For Research Use Only. Not Intended for Diagnostic Or Therapeutic Use.

Product Description
G-15 is a selective antagonist of GPR30 receptor, an estradiol binding receptor that contributes to both uterine and neurological responses. G-15 is reported to oppose the physiological effects of estrogen and inhibit calcium mobilization in vitro.

Specific Protocols

>>	Western Blotting Protocol	>>	Immunoprecipitation Protocol
>>	Immunohistochemistry Protocol	>>	Immunofluorescence Protocol
>>	Immunocytochemistry Protocol	>>	Flow Cytometry Protocol
>>	ChIP Protocol	>>	ELISA Protocol
>>	HPLC Protocol	>>	PCR Protocol