Mirogabalin (CAS: 1138245-13-2 )
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SKU-Pack Size | Availability | Size | Price | |
EBC51031-1MG | In Stock | 1mg | ¥690.00 | |
EBC51031-5MG | In Stock | 5mg | ¥1290.00 | |
EBC51031-10MG | In Stock | 10mg | ¥1990.00 | |
EBC51031-25MG | In Stock | 25mg | ¥3790.00 | |
EBC51016-50MG | In Stock | 50mg | ¥5690.00 |
Please Select The Country You Are In To Find Your Local Distributor. |
北京美瑞克生物科技有限公司 | Phone: +86 010-62890160 / 13691184142(微信同号) | |
2 / F, 128 malianwa North Road, Haidian District, | E-mail: mrkbio@163.com | |
China | Beijing China | Website: www.mrkbio.com |
Product Information | |||||||||||||||||||||
Synonym(s) | DS 5565,DS-5565,DS5565 | ||||||||||||||||||||
Application | Mirogabalin is a calcium channel blocker with analgesic effects | ||||||||||||||||||||
CAS Number | 1138245-13-2 | ||||||||||||||||||||
Purity | ≥99.0% | ||||||||||||||||||||
Molecular Weight | 209.28 | ||||||||||||||||||||
Molecular Formula | C12H19NO2 | ||||||||||||||||||||
SMILES | O=C(O)C[C@]1(CN)[C@]2([H])C=C(CC)C[C@]2([H])C1 | ||||||||||||||||||||
Target & IC50 | α2δ calcium channels | ||||||||||||||||||||
Solubility | H2O: 7.71 mg/mL (36.84 mM) DMSO: 16 mg/mL (76.45 mM)) Methanol: 16 mg/mL (76.45 mM) |
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Preparing Stock Solutions |
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Shipping | Gel Pack | ||||||||||||||||||||
Storage | Store at -20°C | ||||||||||||||||||||
Research Use | For Research Use Only. Not Intended for Diagnostic Or Therapeutic Use. |
Product Description | |
Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the central nervous system (CNS). |
Specific Protocols | |