United Kingdom|
Mirogabalin (CAS: 1138245-13-2 )
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| SKU-Pack Size | Availability | Size | Price | |
| EBC51031-1MG | In Stock | 1mg | £75.90 | |
| EBC51031-5MG | In Stock | 5mg | £141.90 | |
| EBC51031-10MG | In Stock | 10mg | £218.90 | |
| EBC51031-25MG | In Stock | 25mg | £416.90 | |
| EBC51016-50MG | In Stock | 50mg | £625.90 |
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| CUlabSciences | Phone:+44 (0) 1232 330008 | |
| Cambridge House St Thomas' Place Ely, | E-mail:sales@culabsciences.co.uk | |
| United Kingdom | Cambridge CB27 9RD UK | Web:www.culabsciences.co.uk |
| Product Information | |||||||||||||||||||||
| Synonym(s) | DS 5565,DS-5565,DS5565 | ||||||||||||||||||||
| Application | Mirogabalin is a calcium channel blocker with analgesic effects | ||||||||||||||||||||
| CAS Number | 1138245-13-2 | ||||||||||||||||||||
| Purity | ≥99.0% | ||||||||||||||||||||
| Molecular Weight | 209.28 | ||||||||||||||||||||
| Molecular Formula | C12H19NO2 | ||||||||||||||||||||
| SMILES | O=C(O)C[C@]1(CN)[C@]2([H])C=C(CC)C[C@]2([H])C1 | ||||||||||||||||||||
| Target & IC50 | α2δ calcium channels | ||||||||||||||||||||
| Solubility | H2O: 7.71 mg/mL (36.84 mM) DMSO: 16 mg/mL (76.45 mM)) Methanol: 16 mg/mL (76.45 mM) |
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| Preparing Stock Solutions |
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| Shipping | Gel Pack | ||||||||||||||||||||
| Storage | Store at -20°C | ||||||||||||||||||||
| Research Use | For Research Use Only. Not Intended for Diagnostic Or Therapeutic Use. | ||||||||||||||||||||
| Product Description | |
Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the central nervous system (CNS). |
| Specific Protocols | |