Other Biochemicals - Mirogabalin (CAS: 1138245-13-2)

Mirogabalin (CAS: 1138245-13-2)

Catalog #：EBC51031

Biological Activity

Synonyms

DS 5565,DS-5565,DS5565

Application

Mirogabalin is a calcium channel blocker with analgesic effects

CAS Number

1138245-13-2

Purity

≥99.0%

Molecular Weight

209.28

Molecular Formula

C12H19NO2

SMILES

O=C(O)C[C@]1(CN)[C@]2([H])C=C(CC)C[C@]2([H])C1

Target & IC50

α2δ calcium channels

Shipping

Gel Pack

Storage

Store at -20°C

Preparing Stock Solutions

Molecular Structure

ConcentrationSolventMass	1 mg	5 mg	10 mg
1 mM	4.7783 ml	23.8914 ml	47.7829 ml
5 mM	0.9557 ml	4.7783 ml	9.5566 ml
10 mM	0.4778 ml	2.3891 ml	4.7783 ml
50 mM	0.0956 ml	0.4778 ml	0.9557 ml

Solubility
H2O: 7.71 mg/mL (36.84 mM) DMSO: 16 mg/mL (76.45 mM)) Methanol: 16 mg/mL (76.45 mM)

Product Description

Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the CNS. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium-channel complexes in the central nervous system (CNS).